Manufactured by:TriBio Science
RUO

BCTC, TRPV1 blocker

Vanilloid receptor I (TRPV1) antagonist, IC 50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable Solutions in DMSO or ethanol may be stord at -20°C for up to 2 months

SKU:
ABM146684-1
Manufacturer SKU
TBI1086-10MG | TBI1086-50MG
Product type
Biochemical Inhibitors
TargetTRPV1 blocker
Purity>98%

Manufacturer provenance

Manufactured by:
TriBio Science
Sold by:
ABMIUM
Fulfilled from:
Manufacturer facility or confirmed fulfilment location

Know who made it. See the evidence. Buy through one marketplace.

Product description

Vanilloid receptor I (TRPV1) antagonist, IC 50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable

Solutions in DMSO or ethanol may be stord at -20°C for up to 2 months

Key facts & specifications
Also known as
4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide
Molecular weight
372.90
Form / buffer
powder
Activity
Vanilloid receptor I (TRPV1) antagonist, IC 50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable.
Molecular formula
C20H25ClN4O
Solubility
Soluble in DMSO (up to 25 mg/ml) or in Ethanol (up to 15 mg/ml).
Technical note
Stability: ≥ 2 years.
Identifiers & database references
Manufacturer SKU
TBI1086-10MG | TBI1086-50MG
CAS number
393514-24-4
Storage, stability & shipping
Storage conditions
RT
Shipped at
4°C
Long-term storage
RT
Compliance & documents
Datasheet
Open datasheet
Frequently asked questions
Who manufactured this product?

This product is manufactured by TriBio Science and sold through ABMIUM without relabelling.

Can ABMIUM ship this product internationally?

ABMIUM supports global orders. Availability, shipping requirements and applicable import arrangements are confirmed before fulfilment where required.

Can I check suitability before ordering?

Yes. Send your target, sample, application and experimental conditions through ABMIUM MATCH or technical support.

Is this product for clinical use?

Unless the listing expressly states otherwise, ABMIUM products are supplied for research use only and are not for diagnostic or therapeutic use.

TriBio Science
£98.00