SC-51089, Prostaglandin E (EP1) antagonist

SC-51089, Prostaglandin E (EP1) antagonist

100%
Manufactured by:TriBio Science
RUO

SC-51089, Prostaglandin E (EP1) antagonist

Prostaglandin E2 (EP1 receptor) antagonist (pA2=6.5, guinea pig ileum muscle strip assay ). Possesses analgesic activity in vivo (rodent ED50= 6.8 mg/kg). Does not inhibit COX1 and does not block PGE1 induced hyperalgesia

SKU:
ABM148715-1
Manufacturer SKU
TBI1135-25MG | TBI1135-5MG
Product type
Biochemical Inhibitors
TargetProstaglandin E (EP1)
Purity>98%

Manufacturer provenance

Manufactured by:
TriBio Science
Sold by:
ABMIUM
Fulfilled from:
Manufacturer facility or confirmed fulfilment location

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Product description

Prostaglandin E2 (EP1 receptor) antagonist (pA2=6.5, guinea pig ileum muscle strip assay ). Possesses analgesic activity in vivo (rodent ED50= 6.8 mg/kg). Does not inhibit COX1 and does not block PGE1 induced hyperalgesia

Key facts & specifications
Also known as
8-Cholrodibenz(Z)[b,f]oxazepine-10(11H)-carboxylic acid 2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide hydrochloride
Molecular weight
459.34
Form / buffer
powder
Activity
Prostaglandin E2 (EP1 receptor) antagonist (pA2=6.5, guinea pig ileum muscle strip assay ). Possesses analgesic activity in vivo (rodent ED50= 6.8 mg/kg). Does not inhibit COX1 and does not block PGE1 induced hyperalgesia.
Molecular formula
C 22 H 19 ClN 4 O 3 · HCl
Solubility
Soluble in DMSO (up to 25 mg/ml) or in Water (up to 25 mg/ml).
Technical note
Stability: ≥ 1 year.
Identifiers & database references
Manufacturer SKU
TBI1135-25MG | TBI1135-5MG
CAS number
146033-02-5
Storage, stability & shipping
Storage conditions
RT
Shipped at
4°C
Long-term storage
RT
Compliance & documents
Datasheet
Open datasheet
Safety data sheet
Open SDS
Frequently asked questions
Who manufactured this product?

This product is manufactured by TriBio Science and sold through ABMIUM without relabelling.

Can ABMIUM ship this product internationally?

ABMIUM supports global orders. Availability, shipping requirements and applicable import arrangements are confirmed before fulfilment where required.

Can I check suitability before ordering?

Yes. Send your target, sample, application and experimental conditions through ABMIUM MATCH or technical support.

Is this product for clinical use?

Unless the listing expressly states otherwise, ABMIUM products are supplied for research use only and are not for diagnostic or therapeutic use.

TriBio Science
£360.00